Comparative Study
doi: 10.1021/jm00147a002.
Stereostructure-activity relationship of opioid agonist and antagonist bivalent ligands. Evidence for bridging between vicinal opioid receptors
- PMID: 2993609
- DOI: 10.1021/jm00147a002
Item in Clipboard
Comparative Study
Stereostructure-activity relationship of opioid agonist and antagonist bivalent ligands. Evidence for bridging between vicinal opioid receptors
J Med Chem.
1985 Sep.
No abstract available
Similar articles
-
10-Ketonaltrexone and 10-ketooxymorphone.J Med Chem. 1985 Jul;28(7):974-6. doi: 10.1021/jm00145a024. J Med Chem. 1985. PMID: 2409281
-
Agonist-antagonist properties of fluorescent opioid probes in the guinea-pig myenteric plexus-longitudinal muscle preparation.Naunyn Schmiedebergs Arch Pharmacol. 1985 Dec;331(4):355-8. doi: 10.1007/BF00500819. Naunyn Schmiedebergs Arch Pharmacol. 1985. PMID: 2419770
-
Opioid agonist and antagonist bivalent ligands as receptor probes.Life Sci. 1982 Sep 20-27;31(12-13):1283-6. doi: 10.1016/0024-3205(82)90362-9. Life Sci. 1982. PMID: 6292615
-
Chemistry of opioid peptides.Br Med Bull. 1983 Jan;39(1):5-10. doi: 10.1093/oxfordjournals.bmb.a071790. Br Med Bull. 1983. PMID: 6301609 Review. No abstract available.
-
Recent developments in the design of receptor specific opioid peptides.Med Res Rev. 1989 Jul-Sep;9(3):343-401. doi: 10.1002/med.2610090306. Med Res Rev. 1989. PMID: 2547125 Review. No abstract available.
Cited by
-
Synthesis and binding affinity of novel mono- and bivalent morphinan ligands for κ, μ, and δ opioid receptors.Bioorg Med Chem. 2011 May 1;19(9):2808-16. doi: 10.1016/j.bmc.2011.03.052. Epub 2011 Mar 26. Bioorg Med Chem. 2011. PMID: 21482470 Free PMC article.
-
Search for the "ideal analgesic" in pain treatment by engineering the mu-opioid receptor.IUBMB Life. 2010 Feb;62(2):103-11. doi: 10.1002/iub.292. IUBMB Life. 2010. PMID: 20039371 Free PMC article. Review.
-
Design and synthesis of a bivalent ligand to explore the putative heterodimerization of the mu opioid receptor and the chemokine receptor CCR5.Org Biomol Chem. 2012 Apr 7;10(13):2633-46. doi: 10.1039/c2ob06801j. Epub 2012 Feb 22. Org Biomol Chem. 2012. PMID: 22354464 Free PMC article.
-
Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series.Proc Natl Acad Sci U S A. 2005 Dec 27;102(52):19208-13. doi: 10.1073/pnas.0506627102. Epub 2005 Dec 19. Proc Natl Acad Sci U S A. 2005. PMID: 16365317 Free PMC article.
-
In vivo characterization of (-)(-)MCL-144 and (+)(-)MCL-193: isomeric, bivalent ligands with mu/kappa agonist properties.Neurochem Res. 2008 Oct;33(10):2142-50. doi: 10.1007/s11064-008-9752-3. Epub 2008 Jun 5. Neurochem Res. 2008. PMID: 18528756 Free PMC article.
Publication types
MeSH terms
Substances
LinkOut - more resources
Other Literature Sources