Review
doi: 10.1038/sj.bjp.0705420.
Epub 2003 Aug 4.
The 'state' of beta-adrenoceptors
Affiliations
- PMID: 12967928
- PMCID: PMC1574015
- DOI: 10.1038/sj.bjp.0705420
Item in Clipboard
Review
The 'state' of beta-adrenoceptors
Br J Pharmacol.
2003 Sep.
No abstract available
Comment on
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Atypical beta-adrenoceptors, different from beta 3-adrenoceptors and probably from the low-affinity state of beta 1-adrenoceptors, relax the rat isolated mesenteric artery.Br J Pharmacol. 2003 Sep;140(1):3-12. doi: 10.1038/sj.bjp.0705421. Epub 2003 Aug 4. Br J Pharmacol. 2003. PMID: 12967929 Free PMC article.
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References
-
- KAUMANN A.J. Is there a third heart β-adrenoceptor. Trends Pharmacol. Sci. 1989;10:316–320. - PubMed
-
- KAUMANN A.J., ENGELHARDT S., HEIN L., MOLENAAR P., LOHSE M. Abolition of (−)-CGP 12177-evoked cardiostimulation in double β1/β2-adrenoceptor knockout mice. Obligatory role of β1-adrenoceptors for putative β4-adrenoceptor pharmacology. Naunyn-Schmiedeberg's Arch. Pharmacol. 2001;363:87–93. - PubMed
-
- KAUMANN A.J., PREITNER F., SARSERO D., MOLENAAR P., REVELLI J.-P., GIACOBINO J.P. (−)-CGP 12177 causes cardiostimulation and binds to cardiac putative β4-adrenoceptors in both wild-type and β3-adrenoceptor knockout mice. Mol. Pharmacol. 1998;53:670–675. - PubMed
-
- KONKAR A.A., ZHAI Y., GRANNEMAN J.G. β1-adrenergic receptors mediate β3-adrenergic-independent effects of CGP 12177 in brown adipose tissue. Mol. Pharmacol. 2000;57:252–258. - PubMed
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